| Bioactivity | [Arg14,Lys15]Nociceptin is a highly potent and selective NOP receptor (ORL1; OP4) agonist, with an EC50 of 1 nM. [Arg14,Lys15]Nociceptin displays high selectivity over opioid receptors, with IC50s of 0.32, 280, >10000 and 1500 nM for NOP, μ, δ and κ receptors, respectively[1]. |
| Invitro | [Arg14,Lys15]Nociceptin is about 30-fold more potent than Nociceptin (NC) and produces longer lasting effects[2]. |
| Name | [Arg14,Lys15]Nociceptin |
| CAS | 236098-40-1 |
| Shortening | FGGFTGARKSARKRKNQ |
| Formula | C82H137N31O22 |
| Molar Mass | 1909.16 |
| Transport | Room temperature in continental US; may vary elsewhere. |
| Storage | Please store the product under the recommended conditions in the Certificate of Analysis. |